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阿斯利康痛风试验药物Lesinurad或可成为重磅炸弹级产品
发布日期: 2014-03-28
   

      随着世界范围内患有痛风群体比例的不断上升,痛风药物市场已经成为各大医药公司想要竞逐的地方。而阿斯利康凭借着其正处于临床三期研究的药物lesinurad有可能在这一领域拔得头筹。根据相关媒体报道,痛风最近几年在西方国家一直呈现上升趋势。以美国为例,2011年约有830万美国人患有痛风,而2012年英国患有痛风的人数比1997年增加了64%。而目前市面上流行的一些痛风药物主要只有已经使用了50年之久的allopurinol和武田药业和Ipsen公司的febuxostat,后一种药物是在2009年被批准上市。但是这些药物并不能改善所有患者的症状。因此,市场目前急需新的治疗痛风药物的出现。

     阿斯利康的lesinurad是一种URAT1受体抑制剂。在最近的临床三期研究中,这种药物相对于上述两种药物能够明显降低血液中尿酸含量,改善痛风症状。一些分析师认为这种药物一旦上市,其销售额能够突破10亿美元。而另一方面,有些研究人员对这种药物的副作用表示关注,在lesinurad的临床二期研究中,研究人员发现lesinurad可能会导致肾脏问题。(生物谷Bioon.com) 

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